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6EU5

Leishmania major N-myristoyltransferase with bound myristoyl-CoA and inhibitor

Functional Information from GO Data
ChainGOidnamespacecontents
A0004379molecular_functionglycylpeptide N-tetradecanoyltransferase activity
A0005737cellular_componentcytoplasm
A0006499biological_processN-terminal protein myristoylation
A0016746molecular_functionacyltransferase activity
A0046872molecular_functionmetal ion binding
Functional Information from PDB Data
site_idAC1
Number of Residues29
Detailsbinding site for residue MYA A 501
ChainResidue
AHIS2
ACYS160
AVAL161
AARG166
AGLU167
ALYS168
AARG169
ALEU170
AALA171
APRO172
ATHR179
AALA3
AVAL182
ATRP188
AALA190
ATYR192
ATHR193
ALEU198
ATYR394
AHOH660
AHOH709
AHOH738
APHE4
ATRP5
AASN69
ATYR70
AVAL71
APHE158
ALEU159

site_idAC2
Number of Residues17
Detailsbinding site for residue BXN A 502
ChainResidue
AVAL71
AASP73
APHE78
APHE80
ATYR82
ATHR193
ATYR207
AHIS209
ASER320
ALEU331
ATYR335
AASN366
AHIS388
AMET410
ALEU411
AHOH652
AHOH688

Functional Information from PROSITE/UniProt
site_idPS00975
Number of Residues9
DetailsNMT_1 Myristoyl-CoA:protein N-myristoyltransferase signature 1. EINFLCvHK
ChainResidueDetails
AGLU155-LYS163

site_idPS00976
Number of Residues7
DetailsNMT_2 Myristoyl-CoA:protein N-myristoyltransferase signature 2. KFGaGDG
ChainResidueDetails
ALYS381-GLY387

224004

PDB entries from 2024-08-21

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