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6ETE

Crystal structure of KDM4D with tetrazolhydrazide compound 5

Functional Information from PDB Data
site_idAC1
Number of Residues4
Detailsbinding site for residue ZN A 401
ChainResidue
ACYS238
AHIS244
ACYS310
ACYS312

site_idAC2
Number of Residues5
Detailsbinding site for residue NI A 402
ChainResidue
AHIS192
AGLU194
AHIS280
ABWK413
AHOH569

site_idAC3
Number of Residues2
Detailsbinding site for residue NI A 403
ChainResidue
AHIS156
AHOH721

site_idAC4
Number of Residues4
Detailsbinding site for residue EDO A 404
ChainResidue
AARG123
ALYS124
ALYS127
AASN128

site_idAC5
Number of Residues8
Detailsbinding site for residue EDO A 405
ChainResidue
ALYS150
AGLN151
ATRP152
AASN153
AHIS156
ALEU157
AHOH550
AHOH704

site_idAC6
Number of Residues3
Detailsbinding site for residue EDO A 406
ChainResidue
ALYS255
AARG263
AHOH539

site_idAC7
Number of Residues5
Detailsbinding site for residue EDO A 407
ChainResidue
APHE118
AARG263
AILE264
ATHR265
AHOH542

site_idAC8
Number of Residues7
Detailsbinding site for residue EDO A 408
ChainResidue
ALYS109
AGLN111
AASN132
ATRP185
ALYS186
ASO4411
AHOH511

site_idAC9
Number of Residues4
Detailsbinding site for residue EDO A 409
ChainResidue
AHIS103
AASN106
AHOH518
AHOH624

site_idAD1
Number of Residues8
Detailsbinding site for residue EDO A 410
ChainResidue
ATYR179
ATYR181
AGLU194
ASER200
AALA292
AASN294
ABWK413
AHOH569

site_idAD2
Number of Residues6
Detailsbinding site for residue SO4 A 411
ChainResidue
APRO113
ALYS124
AASN128
ATRP185
ALYS186
AEDO408

site_idAD3
Number of Residues6
Detailsbinding site for residue SO4 A 412
ChainResidue
AARG60
AGLU61
ATHR62
AHOH503
AHOH523
AHOH851

site_idAD4
Number of Residues13
Detailsbinding site for residue BWK A 413
ChainResidue
ATYR181
AHIS192
AGLU194
ASER200
AASN202
ALYS210
ATRP212
AHIS280
AALA292
ANI402
AEDO410
AHOH569
AHOH580

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues4
DetailsBINDING: BINDING => ECO:0000250|UniProtKB:B2RXH2
ChainResidueDetails
ATYR136
AASN202
ALYS210
ALYS245

site_idSWS_FT_FI2
Number of Residues3
DetailsBINDING: BINDING => ECO:0000255|PROSITE-ProRule:PRU00538, ECO:0000305|PubMed:26741168
ChainResidueDetails
AHIS192
AGLU194
AHIS280

site_idSWS_FT_FI3
Number of Residues4
DetailsBINDING: BINDING => ECO:0007744|PDB:5F5A, ECO:0007744|PDB:5F5C
ChainResidueDetails
ACYS238
AHIS244
ACYS310
ACYS312

site_idSWS_FT_FI4
Number of Residues2
DetailsMOD_RES: PolyADP-ribosyl glutamic acid => ECO:0000269|PubMed:23102699
ChainResidueDetails
AGLU26
AGLU27

218853

PDB entries from 2024-04-24

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