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6EL6

Glucocorticoid Receptor in complex with compound 4

Functional Information from PDB Data
site_idAC1
Number of Residues7
Detailsbinding site for residue EDO A 801
ChainResidue
APRO541
AALA574
ATRP577
ALEU603
ALYS667
AHOH953
AHOH954

site_idAC2
Number of Residues16
Detailsbinding site for residue B9Q A 802
ChainResidue
ALEU566
AGLY567
AGLN570
AMET601
AMET604
AALA607
ALEU608
AARG611
APHE623
AGLN642
AMET646
ATYR735
ACYS736
ATHR739
ALEU563
AASN564

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues165
DetailsRegion: {"description":"Interaction with CRY1","evidences":[{"source":"PubMed","id":"22170608","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues2
DetailsCross-link: {"description":"Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO)","evidences":[{"source":"PubMed","id":"12144530","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues4
DetailsMotif: {"description":"LXXLL motif 3"}
ChainResidueDetails

246031

PDB entries from 2025-12-10

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