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6EK6

Crystal structure of KDM5B in complex with S49195a.

Functional Information from PDB Data
site_idAC1
Number of Residues4
Detailsbinding site for residue ZN A 801
ChainResidue
ACYS692
ACYS695
ACYS715
AHIS718

site_idAC2
Number of Residues6
Detailsbinding site for residue MN A 802
ChainResidue
AHOH937
ALEU90
AASN91
ALEU413
ATHR416
AGLU419

site_idAC3
Number of Residues5
Detailsbinding site for residue NI A 803
ChainResidue
AHIS499
AGLU501
AHIS587
A90V804
AHOH938

site_idAC4
Number of Residues14
Detailsbinding site for residue 90V A 804
ChainResidue
ATYR425
ATYR488
ASER495
APHE496
AHIS499
AGLU501
ALYS517
AHIS587
AASN591
AALA599
AASN601
ANI803
AHOH938
AHOH1035

site_idAC5
Number of Residues7
Detailsbinding site for residue DMS A 805
ChainResidue
AILE500
ATRP504
AHIS617
ALEU621
AHOH928
AHOH955
AHOH1020

site_idAC6
Number of Residues4
Detailsbinding site for residue DMS A 806
ChainResidue
AARG666
ASER677
ATHR737
AEDO813

site_idAC7
Number of Residues3
Detailsbinding site for residue DMS A 807
ChainResidue
AHIS622
AHIS718
AHOH1041

site_idAC8
Number of Residues6
Detailsbinding site for residue DMS A 808
ChainResidue
AVAL398
AVAL398
AHIS399
AHOH910
AHOH910
AHOH1066

site_idAC9
Number of Residues8
Detailsbinding site for residue EDO A 809
ChainResidue
AVAL615
ATYR618
AARG619
AARG623
ACYS625
ACYS695
ALYS696
ATHR697

site_idAD1
Number of Residues6
Detailsbinding site for residue EDO A 810
ChainResidue
AASP630
ACYS699
APHE700
AMET701
ASER702
AHOH947

site_idAD2
Number of Residues3
Detailsbinding site for residue EDO A 811
ChainResidue
ASER495
APHE496
ACYS497

site_idAD3
Number of Residues4
Detailsbinding site for residue EDO A 812
ChainResidue
AARG612
AASP630
AMET658
AGLU662

site_idAD4
Number of Residues5
Detailsbinding site for residue EDO A 813
ChainResidue
AVAL674
AILE675
ADMS806
AHOH912
AHOH917

site_idAD5
Number of Residues1
Detailsbinding site for residue EDO A 814
ChainResidue
AARG679

site_idAD6
Number of Residues7
Detailsbinding site for residue EDO A 815
ChainResidue
AASP688
AGLU689
AARG690
AGLN691
AVAL693
AGLY711
ALEU713

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues52
DetailsZN_FING: C5HC2 => ECO:0000269|PubMed:26741168, ECO:0000269|PubMed:27214403, ECO:0000269|PubMed:28262558
ChainResidueDetails
ACYS692-MET744

site_idSWS_FT_FI2
Number of Residues4
DetailsBINDING: BINDING => ECO:0000250|UniProtKB:P29375
ChainResidueDetails
ATYR425
ASER507
AASN509
ALYS517

site_idSWS_FT_FI3
Number of Residues3
DetailsBINDING: BINDING => ECO:0000305|PubMed:26741168, ECO:0000305|PubMed:27214403, ECO:0000305|PubMed:28262558
ChainResidueDetails
AHIS499
AGLU501
AHIS587

220113

PDB entries from 2024-05-22

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