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6EJ0

Crystal structure of KDM5B in complex with KDOPZ000049a.

Functional Information from PDB Data
site_idAC1
Number of Residues4
Detailsbinding site for residue ZN A 801
ChainResidue
ACYS692
ACYS695
ACYS715
AHIS718

site_idAC2
Number of Residues6
Detailsbinding site for residue MN A 802
ChainResidue
AHOH909
ALEU90
AASN91
ALEU413
ATHR416
AGLU419

site_idAC3
Number of Residues6
Detailsbinding site for residue EDO A 803
ChainResidue
AASP630
ACYS699
APHE700
AMET701
ASER702
AHOH938

site_idAC4
Number of Residues3
Detailsbinding site for residue EDO A 804
ChainResidue
AGLY524
ATYR525
AARG584

site_idAC5
Number of Residues7
Detailsbinding site for residue DMS A 805
ChainResidue
AILE500
ATRP504
AGLU531
AARG584
AHIS617
ATYR618
AARG623

site_idAC6
Number of Residues8
Detailsbinding site for residue DMS A 806
ChainResidue
ATRP486
ATYR488
AGLU501
ASER507
AALA599
AVAL600
AASN601
AHOH975

site_idAC7
Number of Residues7
Detailsbinding site for residue DMS A 807
ChainResidue
APHE83
AGLY426
AALA427
AASP428
APHE434
ALEU487
AHOH1017

site_idAC8
Number of Residues4
Detailsbinding site for residue DMS A 808
ChainResidue
AGLU631
ALYS635
AGLU683
ATYR736

site_idAC9
Number of Residues3
Detailsbinding site for residue DMS A 809
ChainResidue
AHIS622
AHIS718
AHOH1031

site_idAD1
Number of Residues6
Detailsbinding site for residue MN A 810
ChainResidue
AHIS499
AGLU501
AHIS587
AB7K811
AHOH926
AHOH975

site_idAD2
Number of Residues17
Detailsbinding site for residue B7K A 811
ChainResidue
AARG86
AARG98
ATYR425
AGLY426
ATRP486
ATYR488
APHE496
AHIS499
AASN509
ALYS517
AHIS587
AASN591
AMN810
AHOH910
AHOH926
AHOH975
AHOH1009

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues52
DetailsZN_FING: C5HC2 => ECO:0000269|PubMed:26741168, ECO:0000269|PubMed:27214403, ECO:0000269|PubMed:28262558
ChainResidueDetails
ACYS692-MET744

site_idSWS_FT_FI2
Number of Residues4
DetailsBINDING: BINDING => ECO:0000250|UniProtKB:P29375
ChainResidueDetails
ALYS517
ATYR425
ASER507
AASN509

site_idSWS_FT_FI3
Number of Residues3
DetailsBINDING: BINDING => ECO:0000305|PubMed:26741168, ECO:0000305|PubMed:27214403, ECO:0000305|PubMed:28262558
ChainResidueDetails
AHIS499
AGLU501
AHIS587

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PDB entries from 2024-05-29

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