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6E6J

BRD2_Bromodomain2 complex with inhibitor 744

Functional Information from PDB Data
site_idAC1
Number of Residues17
Detailsbinding site for residue HWV A 501
ChainResidue
ATRP370
APRO430
AVAL435
AHOH611
AHOH616
AHOH640
BTRP370
BMET438
BHWV501
APRO371
APHE372
APRO375
AVAL376
AASP377
ALEU381
ALEU383
AASN429

site_idAC2
Number of Residues14
Detailsbinding site for residue HWV B 501
ChainResidue
ATRP370
AHWV501
BTRP370
BPRO371
BPHE372
BPRO375
BVAL376
BASP377
BLEU383
BASN429
BPRO430
BVAL435
BHOH606
BHOH629

site_idAC3
Number of Residues15
Detailsbinding site for residue HWV C 501
ChainResidue
CTRP370
CPRO371
CPHE372
CVAL376
CASP377
CLEU381
CLEU383
CCYS425
CASN429
CPRO430
CVAL435
CHOH609
CHOH623
DTRP370
DHWV501

site_idAC4
Number of Residues15
Detailsbinding site for residue HWV D 501
ChainResidue
CTRP370
CMET438
CHWV501
DTRP370
DPRO371
DPRO375
DVAL376
DASP377
DLEU381
DLEU383
DASN429
DVAL435
DHOH604
DHOH616
DHOH619

site_idAC5
Number of Residues11
Detailsbinding site for residue HWV E 501
ChainResidue
ETRP370
EPRO371
EPRO375
EVAL376
EASP377
ELEU381
EASN429
EHIS433
EVAL435
FTRP370
FHWV501

site_idAC6
Number of Residues12
Detailsbinding site for residue HWV F 501
ChainResidue
ETRP370
EASP434
EHWV501
FTRP370
FPRO371
FVAL376
FASP377
FLEU381
FLEU383
FASN429
FVAL435
FHOH605

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFykpvDasalglhDYHdiIkhpMdlstVkrkmenrd..Yrdaqefaadvrl.MfsNCykY
ChainResidueDetails
AALA369-TYR428

222415

PDB entries from 2024-07-10

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