6E53
Structure of TERT in complex with a novel telomerase inhibitor
Functional Information from GO Data
Chain | GOid | namespace | contents |
A | 0000781 | cellular_component | chromosome, telomeric region |
A | 0003677 | molecular_function | DNA binding |
A | 0003721 | molecular_function | telomerase RNA reverse transcriptase activity |
A | 0003964 | molecular_function | RNA-directed DNA polymerase activity |
A | 0005634 | cellular_component | nucleus |
A | 0005694 | cellular_component | chromosome |
A | 0006278 | biological_process | RNA-templated DNA biosynthetic process |
A | 0043231 | cellular_component | intracellular membrane-bounded organelle |
A | 0046872 | molecular_function | metal ion binding |
A | 0071897 | biological_process | DNA biosynthetic process |
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 4 |
Details | binding site for residue MG A 601 |
Chain | Residue |
A | ASP251 |
A | ILE252 |
A | ASP343 |
A | HUV603 |
site_id | AC2 |
Number of Residues | 5 |
Details | binding site for residue MG A 602 |
Chain | Residue |
A | ASP251 |
A | ASP343 |
A | ASP344 |
A | HUV603 |
E | DA23 |
site_id | AC3 |
Number of Residues | 19 |
Details | binding site for residue HUV A 603 |
Chain | Residue |
A | LEU141 |
A | ILE187 |
A | LYS189 |
A | ARG194 |
A | ILE196 |
A | ASP251 |
A | ILE252 |
A | ARG253 |
A | ASP254 |
A | ALA255 |
A | TYR256 |
A | GLN308 |
A | GLY309 |
A | ASP343 |
A | LYS372 |
A | MG601 |
A | MG602 |
E | U2 |
E | DA23 |