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6DBH

Crystal structure of PPAR gamma in complex with NMP422

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
B0003677molecular_functionDNA binding
B0004879molecular_functionnuclear receptor activity
B0005634cellular_componentnucleus
B0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues13
Detailsbinding site for residue G3S A 501
ChainResidue
AHIS266
AILE341
ASER342
AMET348
ALYS367
AILE281
AGLY284
ACYS285
AARG288
ASER289
AALA292
AILE326
ALEU333

site_idAC2
Number of Residues2
Detailsbinding site for residue CL A 502
ChainResidue
AARG288
AGLU291

site_idAC3
Number of Residues13
Detailsbinding site for residue G3S B 501
ChainResidue
BLYS263
BILE281
BGLY284
BCYS285
BARG288
BSER289
BILE326
BMET329
BILE341
BSER342
BMET364
BLYS367
BCL503

site_idAC4
Number of Residues2
Detailsbinding site for residue CL B 502
ChainResidue
BLEU228
BMET329

site_idAC5
Number of Residues2
Detailsbinding site for residue CL B 503
ChainResidue
BARG288
BG3S501

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues265
DetailsDomain: {"description":"NR LBD","evidences":[{"source":"PROSITE-ProRule","id":"PRU01189","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues8
DetailsMotif: {"description":"9aaTAD","evidences":[{"source":"PubMed","id":"30468856","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues12
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"9744270","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"2PRG","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI4
Number of Residues4
DetailsCross-link: {"description":"Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in ubiquitin)","evidences":[{"source":"PubMed","id":"36737649","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

242500

PDB entries from 2025-10-01

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