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6D8X

PPAR gamma LBD complexed with the agonist GW1929

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues14
Detailsbinding site for residue EDK A 501
ChainResidue
APHE282
AMET364
AHIS449
ATYR473
AHOH703
AHOH706
AGLY284
ACYS285
ASER289
AHIS323
ATYR327
ALEU330
AILE341
APHE363

site_idAC2
Number of Residues9
Detailsbinding site for residue FLC A 502
ChainResidue
ALYS216
AARG234
ATHR238
AASN375
AHOH606
AHOH640
AHOH644
AHOH690
AHOH726

site_idAC3
Number of Residues5
Detailsbinding site for residue NA A 503
ChainResidue
AARG443
AGLN444
ANA504
AHOH655
AHOH763

site_idAC4
Number of Residues3
Detailsbinding site for residue NA A 504
ChainResidue
ATHR440
AGLN444
ANA503

site_idAC5
Number of Residues2
Detailsbinding site for residue NA A 505
ChainResidue
ALYS457
ATYR473

site_idAC6
Number of Residues7
Detailsbinding site for residue GOL A 506
ChainResidue
APRO227
ALEU228
AARG288
AGLU295
AHOH601
AHOH633
AHOH717

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues265
DetailsDomain: {"description":"NR LBD","evidences":[{"source":"PROSITE-ProRule","id":"PRU01189","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues8
DetailsMotif: {"description":"9aaTAD","evidences":[{"source":"PubMed","id":"30468856","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues6
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"9744270","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"2PRG","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI4
Number of Residues2
DetailsCross-link: {"description":"Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in ubiquitin)","evidences":[{"source":"PubMed","id":"36737649","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

243083

PDB entries from 2025-10-15

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