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6C42

Estrogen Receptor Alpha Ligand Binding Domain in Complex with OP1156

Replaces:  5UF9
Functional Information from PDB Data
site_idAC1
Number of Residues12
Detailsbinding site for residue 85M A 601
ChainResidue
ALEU346
AGLY521
AHIS524
AVAL533
ATHR347
ALEU349
AALA350
AASP351
AGLU353
APHE404
AMET421
AILE424

site_idAC2
Number of Residues11
Detailsbinding site for residue 85M B 601
ChainResidue
BLEU346
BTHR347
BALA350
BASP351
BGLU353
BTRP383
BPHE404
BILE424
BGLY521
BHIS524
BVAL533

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues6
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"9338790","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"9600906","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"1A52","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"1ERE","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues2
DetailsModified residue: {"description":"Phosphotyrosine; by Tyr-kinases","evidences":[{"source":"PubMed","id":"7539106","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues2
DetailsLipidation: {"description":"S-palmitoyl cysteine","evidences":[{"evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

239803

PDB entries from 2025-08-06

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