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6BRW

JAK2 JH2 in complex with XMU-MP-1

Functional Information from GO Data
ChainGOidnamespacecontents
A0004672molecular_functionprotein kinase activity
A0005524molecular_functionATP binding
A0006468biological_processprotein phosphorylation
Functional Information from PDB Data
site_idAC1
Number of Residues14
Detailsbinding site for residue 5BS A 901
ChainResidue
ALEU551
ASER633
ALYS677
AASN678
ALEU680
ASER698
ALEU579
ALYS581
AGLN626
AGLU627
APHE628
AVAL629
ALYS630
AGLY632

site_idAC2
Number of Residues2
Detailsbinding site for residue GOL A 902
ChainResidue
AILE682
AARG683

site_idAC3
Number of Residues4
Detailsbinding site for residue ACT A 903
ChainResidue
AASN673
AARG715
ATRP718
AHOH1060

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsSITE: Breakpoint for translocation to form PCM1-JAK2 fusion protein
ChainResidueDetails
AASP710

site_idSWS_FT_FI2
Number of Residues1
DetailsMOD_RES: Phosphotyrosine => ECO:0007744|PubMed:23186163
ChainResidueDetails
ATYR570

221051

PDB entries from 2024-06-12

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