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6BPI

Crystal structure of SETDB1 Tudor domain with aryl triazole fragment peptide conjugates

Functional Information from PDB Data
site_idAC1
Number of Residues8
Detailsbinding site for residue SO4 A 501
ChainResidue
ALYS229
ALEU241
ALEU242
ASER243
AHIS246
AEDO506
AHOH633
AHOH726

site_idAC2
Number of Residues5
Detailsbinding site for residue SO4 A 502
ChainResidue
ALYS215
AHOH625
AHOH629
AHOH653
AHIS214

site_idAC3
Number of Residues4
Detailsbinding site for residue SO4 A 503
ChainResidue
AARG203
AASP250
ALYS383
AHOH627

site_idAC4
Number of Residues2
Detailsbinding site for residue SO4 A 504
ChainResidue
AARG384
BMLY1

site_idAC5
Number of Residues8
Detailsbinding site for residue EDO A 505
ChainResidue
ATYR193
ASER262
APRO316
ATHR320
AHOH630
AHOH631
AHOH677
AHOH689

site_idAC6
Number of Residues7
Detailsbinding site for residue EDO A 506
ChainResidue
ALYS207
ALYS208
AARG209
ALYS211
AHIS246
ASO4501
AHOH667

site_idAC7
Number of Residues7
Detailsbinding site for residue EDO A 507
ChainResidue
AGLU322
AARG330
ALEU348
ALYS349
AVAL370
AHOH657
AHOH659

site_idAC8
Number of Residues14
Detailsbinding site for Ligand E2G B 4 bound to THR B 3
ChainResidue
AGLY300
AALA302
ACYS329
APHE332
AGLU386
ATRP387
AILE388
ATYR389
ASER392
AARG394
AHOH636
BSER2
BTHR3
BHOH102

224572

PDB entries from 2024-09-04

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