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6B0F

ESTROGEN RECEPTOR ALPHA LIGAND BINDING DOMAIN IN COMPLEX WITH LSZ102

Functional Information from PDB Data
site_idAC1
Number of Residues18
Detailsbinding site for residue C6V A 601
ChainResidue
ALEU346
APHE425
ALEU428
AGLY521
AHIS524
ALEU525
ATYR526
ALYS531
AASN532
AVAL533
ATHR347
ALEU349
AGLU353
ALEU387
AARG394
APHE404
AMET421
AILE424

site_idAC2
Number of Residues3
Detailsbinding site for residue GOL A 602
ChainResidue
AGLU323
APRO325
AARG394

site_idAC3
Number of Residues4
Detailsbinding site for residue GOL A 603
ChainResidue
AGLN441
AGLU444
AALA493
AARG503

site_idAC4
Number of Residues12
Detailsbinding site for residue C6V B 601
ChainResidue
BMET343
BLEU346
BTHR347
BGLU353
BLEU387
BARG394
BPHE404
BILE424
BPHE425
BLEU428
BGLY521
BHIS524

site_idAC5
Number of Residues8
Detailsbinding site for residue GOL B 602
ChainResidue
ALEU327
AARG352
AHIS356
BLEU327
BTYR328
BARG352
BHIS356
BHOH702

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues6
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"9338790","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"9600906","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"1A52","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"1ERE","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues1
DetailsModified residue: {"description":"Phosphotyrosine; by Tyr-kinases","evidences":[{"source":"PubMed","id":"7539106","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues2
DetailsLipidation: {"description":"S-palmitoyl cysteine","evidences":[{"evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

239803

PDB entries from 2025-08-06

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