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6ALB

CREBBP bromodomain in complex with Cpd 30 (1-(3-(3-(1-methyl-1H-pyrazol-4-yl)isoquinolin-8-yl)-1-(tetrahydro-2H-pyran-4-yl)-1,4,6,7-tetrahydro-5H-pyrazolo[4,3-c]pyridin-5-yl)ethan-1-one)

Functional Information from GO Data
ChainGOidnamespacecontents
A0004402molecular_functionhistone acetyltransferase activity
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues4
Detailsbinding site for residue ZN A 1401
ChainResidue
ACYS1199
ACYS1200
AHIS1291
ACYS1294

site_idAC2
Number of Residues4
Detailsbinding site for residue ZN A 1402
ChainResidue
ACYS1283
ACYS1286
ACYS1308
ACYS1311

site_idAC3
Number of Residues4
Detailsbinding site for residue ZN A 1403
ChainResidue
ACYS1219
ACYS1237
ACYS1240
ACYS1213

site_idAC4
Number of Residues5
Detailsbinding site for residue B3P A 1404
ChainResidue
AASN1162
ATRP1165
ATYR1204
AASP1273
ALEU1275

site_idAC5
Number of Residues6
Detailsbinding site for residue BKJ A 1405
ChainResidue
ALEU1109
APRO1110
AGLN1113
AASN1168
APHE1177
AHOH1522

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. SlpFrqpvDpqllgipDYFdiVknpMdlstIkrkldtgq..Yqepwqyvddvwl.MfnNAwlY
ChainResidueDetails
ASER1108-TYR1167

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsMOD_RES: N6-acetyllysine => ECO:0007744|PubMed:19608861
ChainResidueDetails
ALYS1216

218853

PDB entries from 2024-04-24

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