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6A5X

FXR-LBD with HNC180 and SRC1

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006355biological_processregulation of DNA-templated transcription
A0032052molecular_functionbile acid binding
A0038183biological_processbile acid signaling pathway
Functional Information from PDB Data
site_idAC1
Number of Residues5
Detailsbinding site for residue SO4 A 501
ChainResidue
AASN271
ALYS275
ASER279
AALA280
AASN354

site_idAC2
Number of Residues3
Detailsbinding site for residue SO4 A 502
ChainResidue
AGLN416
APHE430
AARG436

site_idAC3
Number of Residues3
Detailsbinding site for residue SO4 A 503
ChainResidue
AGLN267
AGLU268
APRO266

site_idAC4
Number of Residues3
Detailsbinding site for residue SO4 A 504
ChainResidue
ALYS338
ATHR378
AGLN379

site_idAC5
Number of Residues15
Detailsbinding site for residue 9R3 A 505
ChainResidue
AARG264
ATHR270
ALEU287
ATHR288
AMET328
APHE329
AARG331
ASER332
AILE335
ASER342
AGLY343
ATYR369
AHIS447
ATRP454
ATRP469

site_idAC6
Number of Residues5
Detailsbinding site for residue SO4 B 801
ChainResidue
ASER453
AVAL456
AASN457
BTYR751
BLYS755

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues4
DetailsBINDING: BINDING => ECO:0007744|PDB:6HL1
ChainResidueDetails
AARG331
ATYR361
ATYR369
AHIS447

site_idSWS_FT_FI2
Number of Residues1
DetailsMOD_RES: Phosphothreonine; by PKC/PRKCZ => ECO:0000305|PubMed:18668687
ChainResidueDetails
ATHR442

site_idSWS_FT_FI3
Number of Residues2
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO1) => ECO:0000305|PubMed:23546875
ChainResidueDetails
ALYS275

219140

PDB entries from 2024-05-01

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