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5ZQR

Tankyrase-2 in complex with compound 40c

Functional Information from GO Data
ChainGOidnamespacecontents
A0003950molecular_functionNAD+ ADP-ribosyltransferase activity
B0003950molecular_functionNAD+ ADP-ribosyltransferase activity
Functional Information from PDB Data
site_idAC1
Number of Residues4
Detailsbinding site for residue ZN A 1201
ChainResidue
ACYS1081
AHIS1084
ACYS1089
ACYS1092

site_idAC2
Number of Residues16
Detailsbinding site for residue 9H9 A 1202
ChainResidue
AHIS1048
ATYR1050
ATYR1060
APHE1061
AALA1062
ASER1068
ATYR1071
AGLY1074
AILE1075
AHOH1308
BGOL1201
AHIS1031
AGLY1032
ASER1033
APRO1034
APHE1035

site_idAC3
Number of Residues7
Detailsbinding site for residue PO4 A 1203
ChainResidue
AARG977
AHIS979
AARG980
AASP981
ALYS1067
AHOH1311
AHOH1335

site_idAC4
Number of Residues8
Detailsbinding site for residue GOL A 1204
ChainResidue
AHIS1031
AILE1039
APHE1044
AASP1045
AHIS1048
AHOH1308
AHOH1318
AHOH1352

site_idAC5
Number of Residues7
Detailsbinding site for residue GOL A 1205
ChainResidue
APRO1082
AVAL1083
ACYS1092
AHIS1093
APHE1110
AHOH1301
BSER1130

site_idAC6
Number of Residues8
Detailsbinding site for residue GOL B 1201
ChainResidue
ALYS996
ATYR1050
AGLY1053
AMET1054
APHE1055
ATYR1071
A9H91202
BGLU1138

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues4
DetailsBINDING: BINDING => ECO:0000250|UniProtKB:O95271
ChainResidueDetails
ACYS1081
AHIS1084
ACYS1089
ACYS1092

222036

PDB entries from 2024-07-03

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