5X74
The crystal Structure PDE delta in complex with compound (R, R)-1g
Functional Information from GO Data
Chain | GOid | namespace | contents |
A | 0005095 | molecular_function | GTPase inhibitor activity |
A | 0005515 | molecular_function | protein binding |
A | 0005737 | cellular_component | cytoplasm |
A | 0005829 | cellular_component | cytosol |
A | 0005856 | cellular_component | cytoskeleton |
A | 0005929 | cellular_component | cilium |
A | 0007601 | biological_process | visual perception |
A | 0016020 | cellular_component | membrane |
A | 0030659 | cellular_component | cytoplasmic vesicle membrane |
A | 0031267 | molecular_function | small GTPase binding |
A | 0031410 | cellular_component | cytoplasmic vesicle |
A | 0042995 | cellular_component | cell projection |
A | 0050953 | biological_process | sensory perception of light stimulus |
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 16 |
Details | binding site for residue JAY A 201 |
Chain | Residue |
A | MET20 |
A | ILE109 |
A | MET117 |
A | ILE129 |
A | THR131 |
A | VAL145 |
A | LEU147 |
A | TYR149 |
A | LEU22 |
A | TRP32 |
A | ILE53 |
A | CYS56 |
A | ARG61 |
A | GLN78 |
A | GLU88 |
A | TRP90 |