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5WHH

Crystal Structure of Bcl-2-related protein A1 in complex with stapled peptide (AQ7)T(0EH)LRRFGD(MK8)INFRQ(NH2)

Functional Information from GO Data
ChainGOidnamespacecontents
A0042981biological_processregulation of apoptotic process
A0043066biological_processnegative regulation of apoptotic process
Functional Information from PDB Data
site_idAC1
Number of Residues2
Detailsbinding site for residue CL A 201
ChainResidue
AARG68
BAQ775

site_idAC2
Number of Residues20
Detailsbinding site for Ligand residues 0EH B 77 through ILE B 85 bound to THR B 76
ChainResidue
ATHR91
APHE148
BAQ775
BTHR76
BARG79
BARG80
BPHE81
BPHE81
BGLY82
BASN86
BPHE87
BHOH101
BHOH105
ASER43
AVAL44
AASN51
AVAL74
AGLU78
AASN85
AARG88

Functional Information from PROSITE/UniProt
site_idPS01080
Number of Residues20
DetailsBH1 Apoptosis regulator, Bcl-2 family BH1 motif signature. EFeDGiiNWGRIVTIFaFEG
ChainResidueDetails
AGLU78-GLY97

site_idPS01258
Number of Residues12
DetailsBH2 Apoptosis regulator, Bcl-2 family BH2 motif signature. WIrqnGGWEnGF
ChainResidueDetails
ATRP133-PHE144

223532

PDB entries from 2024-08-07

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