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5WFD

Humanized mutant of the Chaetomium thermophilum Polycomb Repressive Complex 2 bound to the inhibitor GSK126

Functional Information from GO Data
ChainGOidnamespacecontents
A0000122biological_processnegative regulation of transcription by RNA polymerase II
A0005634cellular_componentnucleus
A0006325biological_processchromatin organization
A0031491molecular_functionnucleosome binding
B0006338biological_processchromatin remodeling
B0042054molecular_functionhistone methyltransferase activity
Functional Information from PDB Data
site_idAC1
Number of Residues4
Detailsbinding site for residue ZN B 8001
ChainResidue
BCYS727
BCYS748
BCYS755
BCYS760

site_idAC2
Number of Residues3
Detailsbinding site for residue ZN B 8002
ChainResidue
BCYS736
BCYS755
BCYS763

site_idAC3
Number of Residues4
Detailsbinding site for residue ZN B 8003
ChainResidue
BCYS736
BCYS746
BCYS727
BCYS729

site_idAC4
Number of Residues4
Detailsbinding site for residue ZN B 8004
ChainResidue
BCYS685
BHIS687
BCYS691
BCYS697

site_idAC5
Number of Residues4
Detailsbinding site for residue ZN B 8005
ChainResidue
BCYS691
BCYS709
BCYS715
BCYS720

site_idAC6
Number of Residues4
Detailsbinding site for residue ZN B 8006
ChainResidue
BCYS685
BCYS699
BCYS709
BCYS713

site_idAC7
Number of Residues4
Detailsbinding site for residue ZN B 8007
ChainResidue
BCYS508
BCYS511
BCYS516
BHIS518

site_idAC8
Number of Residues4
Detailsbinding site for residue ZN B 8008
ChainResidue
BCYS570
BCYS574
BCYS615
BCYS625

site_idAC9
Number of Residues10
Detailsbinding site for residue A9G B 8009
ChainResidue
BILE302
BTYR303
BTYR304
BHIS307
BGLY808
BTYR809
BARG843
BARG877
BTYR878
BASN880

224931

PDB entries from 2024-09-11

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