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5W1Y

SETD8 in complex with a covalent inhibitor

Functional Information from GO Data
ChainGOidnamespacecontents
A0042799molecular_functionhistone H4K20 methyltransferase activity
B0042799molecular_functionhistone H4K20 methyltransferase activity
Functional Information from PDB Data
site_idAC1
Number of Residues7
Detailsbinding site for residue 9SV A 401
ChainResidue
ATYR303
AASP306
ATHR309
AGLY310
ACYS311
AHOH501
B9SV401

site_idAC2
Number of Residues12
Detailsbinding site for Di-peptide 9SV B 401 and CYS B 311
ChainResidue
BTYR303
BASP306
BTHR309
BGLY310
BTYR312
BMET313
BARG380
BHOH504
BHOH531
BHOH538
ACYS311
A9SV401

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues242
DetailsDomain: {"description":"SET","evidences":[{"source":"PROSITE-ProRule","id":"PRU00190","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues8
DetailsBinding site: {}
ChainResidueDetails

249697

PDB entries from 2026-02-25

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