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5W1Y

SETD8 in complex with a covalent inhibitor

Functional Information from GO Data
ChainGOidnamespacecontents
A0042799molecular_functionhistone H4K20 methyltransferase activity
B0042799molecular_functionhistone H4K20 methyltransferase activity
Functional Information from PDB Data
site_idAC1
Number of Residues7
Detailsbinding site for residue 9SV A 401
ChainResidue
ATYR303
AASP306
ATHR309
AGLY310
ACYS311
AHOH501
B9SV401

site_idAC2
Number of Residues12
Detailsbinding site for Di-peptide 9SV B 401 and CYS B 311
ChainResidue
BTYR303
BASP306
BTHR309
BGLY310
BTYR312
BMET313
BARG380
BHOH504
BHOH531
BHOH538
ACYS311
A9SV401

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues6
DetailsBINDING:
ChainResidueDetails
AASN339
BLYS267
BTYR312
BASN339
ALYS267
ATYR312

219140

PDB entries from 2024-05-01

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