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5TWX

Crystal Structure of BRD9 bromodomain

Functional Information from PDB Data
site_idAC1
Number of Residues14
Detailsbinding site for residue 7P7 B 4000
ChainResidue
BPHE160
BTYR222
DGLN153
DARG154
DPRO157
DPHE163
BPHE161
BVAL165
BILE169
BALA170
BTYR215
BASN216
BARG217
BTHR220

site_idAC2
Number of Residues11
Detailsbinding site for residue 7P7 D 4000
ChainResidue
BTHR166
BALA168
BILE169
CMET175
DPHE160
DILE169
DTYR215
DASN216
DARG217
DTHR220
DTYR222

site_idAC3
Number of Residues29
Detailsbinding site for residues 7P7 A 4000 and 7P7 C 4000
ChainResidue
ALYS155
APRO157
AHIS158
APHE160
APHE160
APHE161
APHE163
AVAL165
AILE169
AALA170
ATYR215
AASN216
AARG217
ATHR220
AVAL221
ATYR222
ATYR222
ALEU225
BMET175
CPHE160
CPHE161
CPHE163
CALA168
CILE169
CALA170
CASN216
CARG217
CTHR220
CTYR222

site_idAC4
Number of Residues29
Detailsbinding site for residues 7P7 A 4000 and 7P7 C 4000
ChainResidue
ALYS155
APRO157
AHIS158
APHE160
APHE160
APHE161
APHE163
AVAL165
AILE169
AALA170
ATYR215
AASN216
AARG217
ATHR220
AVAL221
ATYR222
ATYR222
ALEU225
BMET175
CPHE160
CPHE161
CPHE163
CALA168
CILE169
CALA170
CASN216
CARG217
CTHR220
CTYR222

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues8
DetailsRegion: {"description":"Histone H4K5ac H4K8ac and histone H4K5bu H4K8bu binding","evidences":[{"source":"PubMed","id":"26365797","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues8
DetailsSite: {"description":"Histone H4K5ac H4K8ac and histone H4K5bu H4K8bu binding","evidences":[{"source":"PubMed","id":"26365797","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

246031

PDB entries from 2025-12-10

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