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5O4S

Crystal structure of the human BRPF1 bromodomain in complex with BZ135

Functional Information from PDB Data
site_idAC1
Number of Residues12
Detailsbinding site for residue 9KW A 801
ChainResidue
AILE652
AHOH915
AHOH931
BLYS639
APHE653
APRO658
AGLU661
AVAL662
ACYS704
ATYR707
AASN708
APHE714

site_idAC2
Number of Residues6
Detailsbinding site for residue NO3 A 802
ChainResidue
AGLU694
ALEU729
AARG733
BASP691
BARG733
BHOH918

site_idAC3
Number of Residues11
Detailsbinding site for residue 9KW B 801
ChainResidue
ALYS639
BILE652
BPRO658
BGLU661
BVAL662
BCYS704
BTYR707
BASN708
BPHE714
BHOH911
BHOH930

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues58
DetailsBROMODOMAIN_1 Bromodomain signature. GniFsepvPlsevp..DYLdhIkkpMdfftMkqnleayr..Ylnfddfeedfnl.IvsNClkY
ChainResidueDetails
AGLY650-TYR707

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues104
DetailsDomain: {"description":"Bromo","evidences":[{"source":"PROSITE-ProRule","id":"PRU00035","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

245663

PDB entries from 2025-12-03

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