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5NSP

Crystal structure of TNKS2 in complex with OD334

Functional Information from GO Data
ChainGOidnamespacecontents
A0003950molecular_functionNAD+ poly-ADP-ribosyltransferase activity
B0003950molecular_functionNAD+ poly-ADP-ribosyltransferase activity
C0003950molecular_functionNAD+ poly-ADP-ribosyltransferase activity
D0003950molecular_functionNAD+ poly-ADP-ribosyltransferase activity
Functional Information from PDB Data
site_idAC1
Number of Residues4
Detailsbinding site for residue ZN A 1201
ChainResidue
ACYS1081
AHIS1084
ACYS1089
ACYS1092

site_idAC2
Number of Residues6
Detailsbinding site for residue SO4 A 1202
ChainResidue
CASN1132
AARG977
AHIS979
AARG980
ALYS1067
AGLN1070

site_idAC3
Number of Residues4
Detailsbinding site for residue BCT A 1203
ChainResidue
AHIS1031
AGLY1032
ATYR1060
ASER1068

site_idAC4
Number of Residues5
Detailsbinding site for residue SO4 C 1201
ChainResidue
AASN990
AARG991
CPRO1160
CGLU1161
CHOH1301

site_idAC5
Number of Residues7
Detailsbinding site for residue GOL C 1202
ChainResidue
CARG1128
CPRO1129
CSER1130
CVAL1131
CVAL1131
CASN1132
CGLY1133

site_idAC6
Number of Residues4
Detailsbinding site for residue ZN B 1201
ChainResidue
BCYS1081
BHIS1084
BCYS1089
BCYS1092

site_idAC7
Number of Residues5
Detailsbinding site for residue SO4 B 1202
ChainResidue
BARG977
BHIS979
BARG980
BLYS1067
BGLN1070

site_idAC8
Number of Residues5
Detailsbinding site for residue SO4 B 1203
ChainResidue
BASN990
BARG991
DPRO1160
DGLU1161
DHOH1201

site_idAC9
Number of Residues17
Detailsbinding site for residue 97E B 1204
ChainResidue
BHIS1031
BGLY1032
BSER1033
BPHE1035
BILE1039
BPHE1044
BASP1045
BHIS1048
BALA1049
BILE1051
BGLY1053
BGLY1058
BILE1059
BTYR1060
BTYR1071
BILE1075
BHOH1313

site_idAD1
Number of Residues3
Detailsbinding site for residue BCT B 1205
ChainResidue
BHIS1031
BGLY1032
BSER1068

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues8
DetailsBINDING: BINDING => ECO:0000250|UniProtKB:O95271
ChainResidueDetails
ACYS1081
AHIS1084
ACYS1089
ACYS1092
BCYS1081
BHIS1084
BCYS1089
BCYS1092

237992

PDB entries from 2025-06-25

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