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5NRW

Crystal structure of the human bromodomain of CREBBP bound to the inhibitor XDM4

Functional Information from GO Data
ChainGOidnamespacecontents
A0004402molecular_functionhistone acetyltransferase activity
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues13
Detailsbinding site for residue 96N A 1201
ChainResidue
ALEU1109
AVAL1174
AHOH1312
AHOH1356
AHOH1402
APRO1110
APHE1111
AVAL1115
ALEU1120
AILE1122
ATYR1167
AASN1168
AARG1173

site_idAC2
Number of Residues4
Detailsbinding site for residue EDO A 1202
ChainResidue
AHOH1304
AHOH1313
AHOH1336
AHOH1376

site_idAC3
Number of Residues7
Detailsbinding site for residue EDO A 1203
ChainResidue
AGLU1088
AARG1091
AASP1124
AASP1127
AARG1140
AHOH1325
AHOH1386

site_idAC4
Number of Residues4
Detailsbinding site for residue EDO A 1204
ChainResidue
ATYR1102
AHOH1301
AHOH1303
AHOH1416

site_idAC5
Number of Residues2
Detailsbinding site for residue EDO A 1205
ChainResidue
AARG1103
AHOH1326

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. SlpFrqpvDpqllgipDYFdiVknpMdlstIkrkldtgq..Yqepwqyvddvwl.MfnNAwlY
ChainResidueDetails
ASER1108-TYR1167

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PDB entries from 2024-10-09

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