Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help

5LSU

Structure of the Epigenetic Oncogene MMSET and inhibition by N-Alkyl Sinefungin Derivatives

Functional Information from GO Data
ChainGOidnamespacecontents
A0005634cellular_componentnucleus
A0042054molecular_functionhistone methyltransferase activity
B0005634cellular_componentnucleus
B0042054molecular_functionhistone methyltransferase activity
Functional Information from PDB Data
site_idAC1
Number of Residues4
Detailsbinding site for residue ZN A 1301
ChainResidue
ACYS1144
ACYS1191
ACYS1193
ACYS1198

site_idAC2
Number of Residues4
Detailsbinding site for residue ZN A 1302
ChainResidue
ACYS1016
ACYS1018
ACYS1026
ACYS1032

site_idAC3
Number of Residues4
Detailsbinding site for residue ZN A 1303
ChainResidue
ACYS1041
ACYS1046
ACYS1052
ACYS1026

site_idAC4
Number of Residues18
Detailsbinding site for residue SAM A 1304
ChainResidue
AARG1073
ATRP1075
ATHR1115
AHIS1116
APHE1117
ATYR1118
AARG1138
APHE1139
AASN1141
AHIS1142
ATYR1179
AASN1186
AVAL1190
ACYS1191
AARG1192
AHOH1447
AHOH1471
AHOH1579

site_idAC5
Number of Residues4
Detailsbinding site for residue ZN B 1301
ChainResidue
BCYS1144
BCYS1191
BCYS1193
BCYS1198

site_idAC6
Number of Residues4
Detailsbinding site for residue ZN B 1302
ChainResidue
BCYS1016
BCYS1018
BCYS1026
BCYS1032

site_idAC7
Number of Residues4
Detailsbinding site for residue ZN B 1303
ChainResidue
BCYS1026
BCYS1041
BCYS1046
BCYS1052

site_idAC8
Number of Residues20
Detailsbinding site for residue SAM B 1304
ChainResidue
BARG1073
BTRP1075
BTHR1115
BHIS1116
BPHE1117
BTYR1118
BARG1138
BPHE1139
BASN1141
BHIS1142
BTYR1179
BASN1186
BVAL1190
BCYS1191
BARG1192
BCYS1193
BHOH1407
BHOH1479
BHOH1492
BHOH1503

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues32
DetailsBINDING: BINDING => ECO:0000269|PubMed:27571355, ECO:0007744|PDB:5LSU
ChainResidueDetails
ACYS1052
ATRP1075
ATHR1115
AASN1141
ACYS1144
AASN1186
ACYS1191
AARG1192
ACYS1193
ACYS1198
BCYS1016
BCYS1018
BCYS1026
BCYS1032
BCYS1041
BCYS1046
BCYS1052
BTRP1075
BTHR1115
BASN1141
BCYS1144
BASN1186
BCYS1191
BARG1192
BCYS1193
BCYS1198
ACYS1016
ACYS1018
ACYS1026
ACYS1032
ACYS1041
ACYS1046

221051

PDB entries from 2024-06-12

PDB statisticsPDBj update infoContact PDBjnumon