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5LGA

Structural analysis and biological activities of BXL0124, a Gemini analog of Vitamin D

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues20
Detailsbinding site for residue 6VH A 501
ChainResidue
ATYR175
ASER306
ATRP314
ACYS316
AALA331
AHIS333
ALEU337
AHIS423
ATYR427
ALEU440
AVAL444
ATYR179
APHE448
ALEU255
ALEU258
AALA259
AVAL262
ASER265
AARG302
ASER303

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues5
DetailsBINDING: BINDING => ECO:0000269|PubMed:17218092, ECO:0000269|PubMed:17346665
ChainResidueDetails
ATYR175
ALEU255
AILE299
AHIS333
AHIS423

218853

PDB entries from 2024-04-24

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