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5L8U

Crystal Structure of BAZ2B bromodomain in complex with 3-amino-2-methylpyridine derivative 5

Functional Information from PDB Data
site_idAC1
Number of Residues7
Detailsbinding site for residue 6RS A 2001
ChainResidue
APRO1888
ATYR1901
APHE1943
AASN1944
AILE1950
APGE2002
AHOH2110

site_idAC2
Number of Residues1
Detailsbinding site for residue PGE A 2002
ChainResidue
A6RS2001

site_idAC3
Number of Residues2
Detailsbinding site for residue PGE A 2003
ChainResidue
APRO1899
ALEU1897

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues58
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFllpvNlklvp..GYKkvIkkpMdfstIreklssgq..Ypnletfaldvrl.VfdNCetF
ChainResidueDetails
AALA1886-PHE1943

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsMOD_RES: Phosphothreonine => ECO:0007744|PubMed:21406692
ChainResidueDetails
ALEU1918

site_idSWS_FT_FI2
Number of Residues1
DetailsMOD_RES: Phosphoserine => ECO:0007744|PubMed:21406692
ChainResidueDetails
ATYR1923

220472

PDB entries from 2024-05-29

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