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5KR7

KDM4C bound to pyrazolo-pyrimidine scaffold

Functional Information from PDB Data
site_idAC1
Number of Residues6
Detailsbinding site for residue FE2 A 401
ChainResidue
AHIS190
AGLU192
AHIS278
A6X9403
AHOH501
AHOH582

site_idAC2
Number of Residues4
Detailsbinding site for residue ZN A 402
ChainResidue
ACYS310
ACYS236
AHIS242
ACYS308

site_idAC3
Number of Residues14
Detailsbinding site for residue 6X9 A 403
ChainResidue
ATYR134
ATYR179
ATHR186
APHE187
AHIS190
AASN200
ALYS208
ATRP210
AHIS278
AASN282
AFE2401
AHOH501
AHOH582
AHOH600

site_idAC4
Number of Residues4
Detailsbinding site for residue CL A 404
ChainResidue
AASN126
ATRP183
AHOH687
BARG112

site_idAC5
Number of Residues6
Detailsbinding site for residue FE2 B 401
ChainResidue
BHIS190
BGLU192
BHIS278
B6X9403
BHOH528
BHOH597

site_idAC6
Number of Residues4
Detailsbinding site for residue ZN B 402
ChainResidue
BCYS236
BHIS242
BCYS308
BCYS310

site_idAC7
Number of Residues12
Detailsbinding site for residue 6X9 B 403
ChainResidue
BTYR134
BPHE187
BHIS190
BASN200
BLYS208
BTRP210
BHIS278
BASN282
BFE2401
BHOH528
BHOH597
BHOH638

site_idAC8
Number of Residues3
Detailsbinding site for residue CL B 404
ChainResidue
AARG112
BASN126
BTRP183

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues6
DetailsBINDING: BINDING => ECO:0000250|UniProtKB:B2RXH2
ChainResidueDetails
ATYR134
ALYS208
ALYS243
BTYR134
BLYS208
BLYS243

site_idSWS_FT_FI2
Number of Residues6
DetailsBINDING:
ChainResidueDetails
AHIS190
AGLU192
AHIS278
BHIS190
BGLU192
BHIS278

site_idSWS_FT_FI3
Number of Residues2
DetailsBINDING: BINDING => ECO:0000250
ChainResidueDetails
AASN200
BASN200

site_idSWS_FT_FI4
Number of Residues8
DetailsBINDING: BINDING => ECO:0000269|PubMed:21914792
ChainResidueDetails
ACYS236
AHIS242
ACYS308
ACYS310
BCYS236
BHIS242
BCYS308
BCYS310

222415

PDB entries from 2024-07-10

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