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5KCO

SETDB1 in complex with an early stage, low affinity fragment candidate modelled at reduced occupancy

Functional Information from PDB Data
site_idAC1
Number of Residues5
Detailsbinding site for residue SO4 A 501
ChainResidue
AHIS214
ALYS215
AHOH612
AHOH634
AHOH639

site_idAC2
Number of Residues5
Detailsbinding site for residue SO4 A 502
ChainResidue
AHOH614
AARG209
ATRP363
ALYS364
AASP381

site_idAC3
Number of Residues8
Detailsbinding site for residue 6RO A 503
ChainResidue
APHE296
AGLY300
AALA302
ASER328
APHE332
ATYR389
ASER392
AHOH655

site_idAC4
Number of Residues4
Detailsbinding site for residue DMS A 551
ChainResidue
ALYS207
ALYS208
ALYS211
AHOH652

site_idAC5
Number of Residues7
Detailsbinding site for residue DMS A 552
ChainResidue
ATRP358
ATRP363
APHE379
AASP382
AARG384
AHOH609
AHOH672

site_idAC6
Number of Residues3
Detailsbinding site for residue DMS A 553
ChainResidue
AGLU190
AASN191
ATHR223

223166

PDB entries from 2024-07-31

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