5II1
Crystal Structure of the fifth bromodomain of human polybromo (PB1) in complex with 1-methylisochromeno[3,4-c]pyrazol-5(3H)-one
Functional Information from GO Data
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 12 |
Details | binding site for residue 6BL A 801 |
Chain | Residue |
A | ILE683 |
A | ILE745 |
A | HOH904 |
A | HOH925 |
A | PHE684 |
A | LEU687 |
A | TYR696 |
A | MET704 |
A | MET731 |
A | ALA735 |
A | TYR738 |
A | ASN739 |
site_id | AC2 |
Number of Residues | 14 |
Details | binding site for residue 6BL B 801 |
Chain | Residue |
B | ILE683 |
B | PHE684 |
B | LEU687 |
B | LEU693 |
B | TYR696 |
B | MET704 |
B | ASP705 |
B | MET731 |
B | ALA735 |
B | TYR738 |
B | ASN739 |
B | ILE745 |
B | HOH906 |
B | HOH908 |
Functional Information from PROSITE/UniProt
site_id | PS00633 |
Number of Residues | 58 |
Details | BROMODOMAIN_1 Bromodomain signature. SaiFlrlpSrselp..DYYltIkkpMdmekIrshmmank..Yqdidsmvedfvm.MfnNActY |
Chain | Residue | Details |
A | SER681-TYR738 |
Functional Information from SwissProt/UniProt
site_id | SWS_FT_FI1 |
Number of Residues | 220 |
Details | Domain: {"description":"Bromo 5","evidences":[{"source":"PROSITE-ProRule","id":"PRU00035","evidenceCode":"ECO:0000255"}]} |
Chain | Residue | Details |
site_id | SWS_FT_FI2 |
Number of Residues | 2 |
Details | Modified residue: {"description":"Phosphoserine","evidences":[{"source":"PubMed","id":"23186163","evidenceCode":"ECO:0007744"}]} |
Chain | Residue | Details |
site_id | SWS_FT_FI3 |
Number of Residues | 4 |
Details | Cross-link: {"description":"Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2)","evidences":[{"source":"PubMed","id":"25755297","evidenceCode":"ECO:0007744"},{"source":"PubMed","id":"28112733","evidenceCode":"ECO:0007744"}]} |
Chain | Residue | Details |