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5GWZ

The structure of Porcine epidemic diarrhea virus main protease in complex with an inhibitor

Functional Information from GO Data
ChainGOidnamespacecontents
A0008233molecular_functionpeptidase activity
A0019082biological_processviral protein processing
B0008233molecular_functionpeptidase activity
B0019082biological_processviral protein processing
Functional Information from PDB Data
site_idAC1
Number of Residues19
DetailsBINDING SITE FOR CHAIN D OF N-[(5-METHYLISOXAZOL-3-YL)CARBONYL]ALANYL-L-VALYL-N~1~- ((1R,2Z)-4-(BENZYLOXY)-4-OXO-1-{[(3R)-2-OXOPYRROLIDIN-3- YL]METHYL}BUT-2-ENYL)-L-LEUCINAMIDE
ChainResidue
AHIS235
BLEU164
BGLU165
BHIS171
BGLN187
BPRO188
BTHR189
BLEU190
BGLN191
BHOH430
DHOH101
BMET25
BALA26
BHIS41
BPHE139
BGLY142
BCYS144
BHIS162
BGLN163

site_idAC2
Number of Residues16
DetailsBINDING SITE FOR CHAIN E OF N-[(5-METHYLISOXAZOL-3-YL)CARBONYL]ALANYL-L-VALYL-N~1~- ((1R,2Z)-4-(BENZYLOXY)-4-OXO-1-{[(3R)-2-OXOPYRROLIDIN-3- YL]METHYL}BUT-2-ENYL)-L-LEUCINAMIDE
ChainResidue
AMET25
ALEU27
AHIS41
APHE139
AASN141
AGLY142
ACYS144
AHIS162
AGLN163
ALEU164
AGLU165
AHIS171
AGLN187
APRO188
ATHR189
ALEU190

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues4
DetailsACT_SITE: For 3CL-PRO activity => ECO:0000255|PROSITE-ProRule:PRU00772, ECO:0000269|PubMed:27173881
ChainResidueDetails
BHIS41
BCYS144
AHIS41
ACYS144

site_idSWS_FT_FI2
Number of Residues2
DetailsSITE: Cleavage; by 3CL-PRO => ECO:0000250
ChainResidueDetails
BGLN302
AGLN302

222926

PDB entries from 2024-07-24

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