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5FRN

Crystal structure of the Prototype Foamy Virus (PFV) intasome in complex with magnesium and the INSTI XZ419 (compound 4c)

Functional Information from GO Data
ChainGOidnamespacecontents
A0003676molecular_functionnucleic acid binding
A0015074biological_processDNA integration
B0003676molecular_functionnucleic acid binding
B0015074biological_processDNA integration
Functional Information from PDB Data
site_idAC1
Number of Residues4
DetailsBINDING SITE FOR RESIDUE ZN A 393
ChainResidue
AHIS62
AHIS66
ACYS96
ACYS99

site_idAC2
Number of Residues5
DetailsBINDING SITE FOR RESIDUE MG A 394
ChainResidue
AASP128
AASP185
AHOH3016
AHOH3017
DQUW1018

site_idAC3
Number of Residues4
DetailsBINDING SITE FOR RESIDUE MG A 395
ChainResidue
AASP128
AGLU221
AHOH3018
DQUW1018

site_idAC4
Number of Residues5
DetailsBINDING SITE FOR RESIDUE SO4 B 393
ChainResidue
BLYS219
BARG222
BSER258
BPRO259
BVAL260

site_idAC5
Number of Residues15
DetailsBINDING SITE FOR RESIDUE QUW D 1018
ChainResidue
AASP128
AASP185
AGLN186
APRO211
ATYR212
APRO214
AGLN215
AGLU221
AMG394
AMG395
AHOH3016
AHOH3017
CDG4
DDC16
DDA17

site_idAC6
Number of Residues3
DetailsBINDING SITE FOR RESIDUE SO4 A 2001
ChainResidue
ASER136
AGLN137
ALYS241

site_idAC7
Number of Residues3
DetailsBINDING SITE FOR RESIDUE SO4 A 2002
ChainResidue
AGLY187
AALA188
DDA17

site_idAC8
Number of Residues5
DetailsBINDING SITE FOR RESIDUE SO4 A 2003
ChainResidue
ALYS228
ASER332
ALEU333
AARG336
AHOH3061

site_idAC9
Number of Residues3
DetailsBINDING SITE FOR RESIDUE SO4 A 2004
ChainResidue
AHIS338
ALYS339
AHIS357

site_idBC1
Number of Residues4
DetailsBINDING SITE FOR RESIDUE GOL A 1376
ChainResidue
ASER162
ATHR163
ASER164
AHOH3024

site_idBC2
Number of Residues5
DetailsBINDING SITE FOR RESIDUE GOL B 1299
ChainResidue
AGLN296
BTYR263
BGLN267
BGLY271
BASP273

site_idBC3
Number of Residues2
DetailsBINDING SITE FOR RESIDUE GOL A 1377
ChainResidue
AASP116
CDT3

site_idBC4
Number of Residues6
DetailsBINDING SITE FOR RESIDUE GOL C 1020
ChainResidue
ATYR303
AGOL1378
CDC6
CDA7
CDT8
DDC11

site_idBC5
Number of Residues5
DetailsBINDING SITE FOR RESIDUE GOL B 1300
ChainResidue
ASER175
BLEU155
BTYR243
BPRO247
BGLN250

site_idBC6
Number of Residues6
DetailsBINDING SITE FOR RESIDUE GOL A 1378
ChainResidue
AARG114
ATYR303
APRO305
AHOH3066
CDC6
CGOL1020

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues4
DetailsBINDING: BINDING => ECO:0000250
ChainResidueDetails
AASP123
AASP185
BASP123
BASP185

221371

PDB entries from 2024-06-19

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