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5FKO

TetR(D) E147A mutant in complex with anhydrotetracycline and magnesium

Functional Information from GO Data
ChainGOidnamespacecontents
A0000976molecular_functiontranscription cis-regulatory region binding
A0003677molecular_functionDNA binding
A0003700molecular_functionDNA-binding transcription factor activity
A0006355biological_processregulation of DNA-templated transcription
A0045892biological_processnegative regulation of DNA-templated transcription
A0046677biological_processresponse to antibiotic
A0046872molecular_functionmetal ion binding
Functional Information from PDB Data
site_idAC1
Number of Residues17
DetailsBINDING SITE FOR RESIDUE TDC A 1209
ChainResidue
AHIS64
AGLN116
ASER138
AMET177
AMG1210
AHOH2065
AHOH2066
AHOH2067
AHOH2073
ASER67
AASN82
APHE86
AHIS100
ATHR103
AARG104
APRO105
AVAL113

site_idAC2
Number of Residues5
DetailsBINDING SITE FOR RESIDUE MG A 1210
ChainResidue
AHIS100
ATDC1209
AHOH2065
AHOH2066
AHOH2067

site_idAC3
Number of Residues3
DetailsBINDING SITE FOR RESIDUE CL A 1211
ChainResidue
AGLY102
AHOH2066
AHOH2087

site_idAC4
Number of Residues4
DetailsBINDING SITE FOR RESIDUE CL A 1212
ChainResidue
ASER2
AARG3
ASER74
ASER77

site_idAC5
Number of Residues4
DetailsBINDING SITE FOR RESIDUE CL A 1213
ChainResidue
ALEU4
AGLN76
AARG80
AHOH2100

site_idAC6
Number of Residues2
DetailsBINDING SITE FOR RESIDUE CL A 1214
ChainResidue
AASN5
AGLU7

site_idAC7
Number of Residues2
DetailsBINDING SITE FOR RESIDUE CL A 1215
ChainResidue
ATHR26
ATHR27

Functional Information from PROSITE/UniProt
site_idPS01081
Number of Residues32
DetailsHTH_TETR_1 TetR-type HTH domain signature. GIdglTTrkLaqklgIEqPtLYwHVkNKralL
ChainResidueDetails
AGLY21-LEU52

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues19
DetailsDNA_BIND: H-T-H motif => ECO:0000255|PROSITE-ProRule:PRU00335
ChainResidueDetails
ATHR26-VAL45

site_idSWS_FT_FI2
Number of Residues3
DetailsBINDING: BINDING => ECO:0000269|PubMed:8153629, ECO:0007744|PDB:2TRT
ChainResidueDetails
AHIS64
AASN82
AHIS100

224572

PDB entries from 2024-09-04

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