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5FG4

Crystal structure of the bromodomain of human BRPF1 in complex with OF-1 chemical probe

Functional Information from PDB Data
site_idAC1
Number of Residues11
Detailsbinding site for residue 5XE A 801
ChainResidue
ALYS639
AHOH905
AHOH938
AILE652
APHE653
AVAL657
APRO658
AGLU661
AVAL662
AASN708
APHE714

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues58
DetailsBROMODOMAIN_1 Bromodomain signature. GniFsepvPlsevp..DYLdhIkkpMdfftMkqnleayr..Ylnfddfeedfnl.IvsNClkY
ChainResidueDetails
AGLY650-TYR707

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues104
DetailsDomain: {"description":"Bromo","evidences":[{"source":"PROSITE-ProRule","id":"PRU00035","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

238895

PDB entries from 2025-07-16

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