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5FFY

Crystal structure of the bromodomain of human BRPF1 in complex with a benzimidazole ligand

Functional Information from PDB Data
site_idAC1
Number of Residues13
Detailsbinding site for residue 5XD A 801
ChainResidue
ALYS639
APHE714
AHOH907
AHOH939
AHOH959
AGLU642
AILE652
APHE653
AVAL657
APRO658
AGLU661
AVAL662
AASN708

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues58
DetailsBROMODOMAIN_1 Bromodomain signature. GniFsepvPlsevp..DYLdhIkkpMdfftMkqnleayr..Ylnfddfeedfnl.IvsNClkY
ChainResidueDetails
AGLY650-TYR707

246031

PDB entries from 2025-12-10

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