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5FDR

Mcl-1 complexed with small molecule inhibitor

Functional Information from GO Data
ChainGOidnamespacecontents
A0042981biological_processregulation of apoptotic process
B0042981biological_processregulation of apoptotic process
C0042981biological_processregulation of apoptotic process
D0042981biological_processregulation of apoptotic process
Functional Information from PDB Data
site_idAC1
Number of Residues16
Detailsbinding site for residue 5X3 A 400
ChainResidue
AHIS224
ATHR266
ALEU267
APHE270
AGLY271
BTHR226
CASP256
CGLY257
AALA227
APHE228
AMET231
AMET250
AVAL253
AASN260
AGLY262
AARG263

site_idAC2
Number of Residues14
Detailsbinding site for residue 5X3 B 400
ChainResidue
AGLY219
AARG222
AASN223
BALA227
BPHE228
BMET231
BVAL249
BMET250
BVAL253
BASP256
BGLY257
BARG263
BLEU267
BPHE270

site_idAC3
Number of Residues15
Detailsbinding site for residue 5X3 C 400
ChainResidue
AASP256
AGLY257
CHIS224
CALA227
CPHE228
CMET231
CMET250
CVAL253
CASN260
CGLY262
CARG263
CTHR266
CLEU267
CPHE270
DTHR226

site_idAC4
Number of Residues16
Detailsbinding site for residue 5X3 D 400
ChainResidue
CGLY219
CARG222
CASN223
DALA227
DPHE228
DMET231
DMET250
DVAL253
DPHE254
DASP256
DGLY257
DARG263
DTHR266
DLEU267
DPHE270
DILE294

Functional Information from PROSITE/UniProt
site_idPS01080
Number of Residues20
DetailsBH1 Apoptosis regulator, Bcl-2 family BH1 motif signature. VFsDGvtNWGRIVTLIsFGA
ChainResidueDetails
AVAL253-ALA272

site_idPS01258
Number of Residues12
DetailsBH2 Apoptosis regulator, Bcl-2 family BH2 motif signature. WLvkqRGWDgFV
ChainResidueDetails
ATRP305-VAL316

site_idPS01259
Number of Residues15
DetailsBH3 Apoptosis regulator, Bcl-2 family BH3 motif signature. AletLRrVGDGVQRN
ChainResidueDetails
AALA209-ASN223

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues12
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in ubiquitin)
ChainResidueDetails
ALYS194
DLYS194
DLYS197
ALYS197
BLYS194
BLYS197
CLYS194
CLYS197

221716

PDB entries from 2024-06-26

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