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5C91

NEDD4 HECT with covalently bound indole-based inhibitor

Functional Information from GO Data
ChainGOidnamespacecontents
A0004842molecular_functionubiquitin-protein transferase activity
Functional Information from PDB Data
site_idAC1
Number of Residues10
Detailsbinding site for residue 4YU A 901
ChainResidue
AGLU554
ALYS747
ATYR604
ATYR605
ALEU607
AASN621
AASN623
ASER624
ACYS627
AASN628

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsActive site: {"description":"Glycyl thioester intermediate","evidences":[{"source":"PROSITE-ProRule","id":"PRU00104","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues2
DetailsCross-link: {"description":"Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in ubiquitin)","evidences":[{"source":"PubMed","id":"32101753","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

247536

PDB entries from 2026-01-14

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