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5AVI

Crystal structure of LXRalpha in complex with tert-butyl benzoate analog, compound 4

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006629biological_processlipid metabolic process
C0003677molecular_functionDNA binding
C0004879molecular_functionnuclear receptor activity
C0006629biological_processlipid metabolic process
Functional Information from PDB Data
site_idAC1
Number of Residues13
Detailsbinding site for residue 4KM A 501
ChainResidue
APHE257
APHE335
AGLN424
ALEU428
ATRP443
ALEU260
AALA261
ASER264
AILE295
ATHR302
AARG305
APHE315
ALEU331

site_idAC2
Number of Residues15
Detailsbinding site for residue 4KM C 501
ChainResidue
CPHE257
CLEU260
CALA261
CSER264
CILE295
CTHR302
CARG305
CPHE315
CLEU331
CPHE335
CHIS421
CGLN424
CLEU428
CLEU435
CTRP443

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsMOD_RES: Phosphoserine => ECO:0007744|PubMed:23186163
ChainResidueDetails
BSER698
DSER698

224201

PDB entries from 2024-08-28

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