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5A7R

Human poly(ADP-ribose) glycohydrolase in complex with synthetic dimeric ADP-ribose

Functional Information from GO Data
ChainGOidnamespacecontents
A0004649molecular_functionpoly(ADP-ribose) glycohydrolase activity
A0005975biological_processcarbohydrate metabolic process
A0006282biological_processregulation of DNA repair
Functional Information from PDB Data
site_idAC1
Number of Residues4
DetailsBINDING SITE FOR RESIDUE BME A 1966
ChainResidue
AASP575
ACYS603
APRO673
AHOH2212

site_idAC2
Number of Residues6
DetailsBINDING SITE FOR RESIDUE SO4 A 1967
ChainResidue
AHOH2041
AILE484
AARG485
AVAL486
AASP487
APHE498

site_idAC3
Number of Residues5
DetailsBINDING SITE FOR RESIDUE SO4 A 1968
ChainResidue
ALYS567
APRO838
AARG842
AHOH2356
AHOH2417

site_idAC4
Number of Residues2
DetailsBINDING SITE FOR RESIDUE SO4 A 1969
ChainResidue
AALA750
AAR61965

site_idAC5
Number of Residues4
DetailsBINDING SITE FOR RESIDUE SO4 A 1970
ChainResidue
AGLU459
AMET461
AARG462
AARG466

site_idAC6
Number of Residues3
DetailsBINDING SITE FOR RESIDUE SO4 A 1971
ChainResidue
AGLU839
ALYS840
AARG843

site_idAC7
Number of Residues6
DetailsBINDING SITE FOR RESIDUE SO4 A 1972
ChainResidue
ATYR564
AARG644
AASN646
AARG941
AHOH2127
AHOH2186

site_idAC8
Number of Residues2
DetailsBINDING SITE FOR RESIDUE SO4 A 1973
ChainResidue
ATRP506
AARG644

site_idAC9
Number of Residues10
DetailsBINDING SITE FOR RESIDUE GOL A 1974
ChainResidue
AGLU727
AGLN735
AARG758
AASN762
AGLN788
ASER809
AHOH2268
AHOH2275
AHOH2314
AHOH2331

site_idBC1
Number of Residues7
DetailsBINDING SITE FOR RESIDUE GOL A 1975
ChainResidue
AGLU709
ACYS711
AGLU712
ATHR924
AASP927
ALYS930
AHOH2418

site_idBC2
Number of Residues5
DetailsBINDING SITE FOR RESIDUE GOL A 1976
ChainResidue
AASN869
ACYS872
AASP904
AAR61964
AHOH2378

site_idBC3
Number of Residues4
DetailsBINDING SITE FOR RESIDUE GOL A 1977
ChainResidue
AALA796
AGLU797
AAR61965
AHOH2325

site_idBC4
Number of Residues7
DetailsBINDING SITE FOR RESIDUE GOL A 1978
ChainResidue
AHIS828
APHE829
AARG830
AARG831
AASP834
ALYS840
AHOH2419

site_idBC5
Number of Residues3
DetailsBINDING SITE FOR RESIDUE GOL A 1979
ChainResidue
AARG685
AALA689
AGLU787

site_idBC6
Number of Residues6
DetailsBINDING SITE FOR RESIDUE GOL A 1980
ChainResidue
AASN508
ALEU614
AGLU652
AHOH2075
AHOH2200
AHOH2420

site_idBC7
Number of Residues6
DetailsBINDING SITE FOR RESIDUE GOL A 1981
ChainResidue
AASN740
AHIS828
APHE875
AAR61965
AHOH2286
AHOH2421

site_idBC8
Number of Residues3
DetailsBINDING SITE FOR RESIDUE GOL A 1982
ChainResidue
AGLU585
ALEU589
AHOH2220

site_idBC9
Number of Residues6
DetailsBINDING SITE FOR RESIDUE GOL A 1983
ChainResidue
AHIS501
ATYR502
APRO605
AASN606
APPI1987
AHOH2062

site_idCC1
Number of Residues5
DetailsBINDING SITE FOR RESIDUE GOL A 1984
ChainResidue
AGLY492
AGLN551
ALYS554
AALA690
AHOH2113

site_idCC2
Number of Residues7
DetailsBINDING SITE FOR RESIDUE PPI A 1985
ChainResidue
AHOH2125
AHOH2195
ATYR521
AARG535
ATYR560
AASN561
AVAL562

site_idCC3
Number of Residues4
DetailsBINDING SITE FOR RESIDUE PPI A 1986
ChainResidue
ALEU471
AARG816
AHOH2235
AHOH2313

site_idCC4
Number of Residues4
DetailsBINDING SITE FOR RESIDUE PPI A 1987
ChainResidue
ACYS515
AGLU517
AGOL1983
AHOH2092

site_idCC5
Number of Residues3
DetailsBINDING SITE FOR RESIDUE PPI A 1988
ChainResidue
AGLY724
APPI1990
AHOH2264

site_idCC6
Number of Residues3
DetailsBINDING SITE FOR RESIDUE PPI A 1989
ChainResidue
ASER655
AARG741
AHOH2199

site_idCC7
Number of Residues6
DetailsBINDING SITE FOR RESIDUE PPI A 1990
ChainResidue
ATHR725
ATYR792
AGLY794
APPI1988
AHOH2318
AHOH2323

site_idCC8
Number of Residues35
DetailsBinding site for residues AR6 A1964 and AR6 A1965
ChainResidue
AARG663
AILE726
AGLU727
APHE738
AASN740
AGLY745
ASER749
AALA750
AGLY751
ALEU752
AVAL753
AGLN754
AGLU755
AASN756
ATYR795
AASN869
AGLY871
ACYS872
AGLY873
AALA874
APHE875
APHE902
ASO41969
AGOL1976
AGOL1977
AGOL1981
AHOH2284
AHOH2285
AHOH2288
AHOH2320
AHOH2325
AHOH2326
AHOH2327
AHOH2365
AHOH2416

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsACT_SITE: ACT_SITE => ECO:0000269|PubMed:23251397
ChainResidueDetails
AASP737

site_idSWS_FT_FI2
Number of Residues2
DetailsACT_SITE: ACT_SITE => ECO:0000269|PubMed:21892188, ECO:0000269|PubMed:23251397
ChainResidueDetails
AGLU755
AASN756

site_idSWS_FT_FI3
Number of Residues4
DetailsBINDING: BINDING => ECO:0000269|PubMed:23251397, ECO:0000269|PubMed:30472116
ChainResidueDetails
AILE726
AASN740
AGLN754
AASN869

site_idSWS_FT_FI4
Number of Residues1
DetailsBINDING: BINDING => ECO:0000250|UniProtKB:Q9QYM2
ChainResidueDetails
ATYR795

site_idSWS_FT_FI5
Number of Residues1
DetailsMOD_RES: Phosphoserine => ECO:0007744|PubMed:23186163
ChainResidueDetails
ASER448

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PDB entries from 2024-05-01

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