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4ZJR

RORgamma in complex with inverse agonist 48

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
B0003677molecular_functionDNA binding
B0004879molecular_functionnuclear receptor activity
B0005634cellular_componentnucleus
B0006355biological_processregulation of DNA-templated transcription
C0003677molecular_functionDNA binding
C0004879molecular_functionnuclear receptor activity
C0005634cellular_componentnucleus
C0006355biological_processregulation of DNA-templated transcription
D0003677molecular_functionDNA binding
D0004879molecular_functionnuclear receptor activity
D0005634cellular_componentnucleus
D0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues12
Detailsbinding site for residue 4P3 A 501
ChainResidue
ATRP317
AILE400
APHE401
AHIS479
ACYS320
AHIS323
ALEU324
APHE378
AGLU379
APHE388
ALEU396
AILE397

site_idAC2
Number of Residues14
Detailsbinding site for residue 4P3 B 501
ChainResidue
BTRP317
BCYS320
BHIS323
BLEU324
BMET365
BVAL376
BPHE378
BGLU379
BPHE388
BLEU396
BILE397
BILE400
BHIS479
BHOH607

site_idAC3
Number of Residues12
Detailsbinding site for residue 4P3 C 501
ChainResidue
CCYS320
CHIS323
CVAL376
CGLU379
CPHE388
CLEU391
CCYS393
CLEU396
CILE397
CILE400
CPHE401
CHIS479

site_idAC4
Number of Residues13
Detailsbinding site for residue 4P3 D 501
ChainResidue
DCYS320
DHIS323
DMET365
DVAL376
DPHE377
DPHE378
DGLU379
DPHE388
DLEU396
DILE397
DILE400
DPHE401
DHIS479

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PDB entries from 2024-07-24

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