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4WPF

Crystal structure of RORc in complex with a phenyl sulfonamide agonist

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
D0003677molecular_functionDNA binding
D0004879molecular_functionnuclear receptor activity
D0005634cellular_componentnucleus
D0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues12
Detailsbinding site for residue 3SN A 601
ChainResidue
AGLN286
AILE397
AILE400
AHOH732
ALEU287
ATRP317
ACYS320
ALEU324
AALA368
APHE378
APHE388
ALEU396

site_idAC2
Number of Residues12
Detailsbinding site for residue 3SN D 601
ChainResidue
DGLN286
DLEU287
DTRP317
DLEU324
DMET365
DALA368
DPHE377
DPHE378
DPHE388
DILE397
DILE400
DHOH738

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues478
DetailsDomain: {"description":"NR LBD","evidences":[{"source":"PROSITE-ProRule","id":"PRU01189","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues10
DetailsMotif: {"description":"AF-2"}
ChainResidueDetails

239149

數據於2025-07-23公開中

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