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4V05

FGFR1 in complex with AZD4547.

Functional Information from GO Data
ChainGOidnamespacecontents
A0004672molecular_functionprotein kinase activity
A0004713molecular_functionprotein tyrosine kinase activity
A0005007molecular_functionfibroblast growth factor receptor activity
A0005524molecular_functionATP binding
A0006468biological_processprotein phosphorylation
B0004672molecular_functionprotein kinase activity
B0004713molecular_functionprotein tyrosine kinase activity
B0005007molecular_functionfibroblast growth factor receptor activity
B0005524molecular_functionATP binding
B0006468biological_processprotein phosphorylation
Functional Information from PDB Data
site_idAC1
Number of Residues7
DetailsBINDING SITE FOR RESIDUE EDO A 1766
ChainResidue
ALYS665
ATRP684
ATYR701
AARG718
AMET719
ATRP737
AHOH2037

site_idAC2
Number of Residues5
DetailsBINDING SITE FOR RESIDUE EDO B 1765
ChainResidue
BASP524
BLEU528
BGLU531
BLYS514
BLEU516

site_idAC3
Number of Residues5
DetailsBINDING SITE FOR RESIDUE EDO B 1766
ChainResidue
BTYR701
BARG718
BMET719
BTRP737
BHOH2043

site_idAC4
Number of Residues5
DetailsBINDING SITE FOR RESIDUE EDO A 1767
ChainResidue
AALA615
AHIS679
ATHR746
APHE747
ALYS748

site_idAC5
Number of Residues3
DetailsBINDING SITE FOR RESIDUE EDO A 1768
ChainResidue
ALYS566
AARG576
A66T1769

site_idAC6
Number of Residues15
DetailsBINDING SITE FOR RESIDUE 66T A 1769
ChainResidue
ALEU484
AALA512
ALYS514
AGLU531
AILE545
AVAL561
AGLU562
ATYR563
AALA564
ASER565
AGLY567
AGLU571
ALEU630
AASP641
AEDO1768

site_idAC7
Number of Residues16
DetailsBINDING SITE FOR RESIDUE 66T B 1767
ChainResidue
BALA512
BLYS514
BMET535
BILE545
BVAL559
BVAL561
BGLU562
BTYR563
BALA564
BSER565
BGLY567
BLEU630
BALA640
BASP641
BPHE642
BHOH2063

site_idAC8
Number of Residues7
DetailsBINDING SITE FOR RESIDUE SO4 A 1770
ChainResidue
AARG570
AARG627
ATHR657
AASN659
AARG661
AHOH2033
AHOH2035

site_idAC9
Number of Residues6
DetailsBINDING SITE FOR RESIDUE SO4 B 1768
ChainResidue
BARG570
BARG627
BTHR657
BASN659
BARG661
BHOH2039

site_idBC1
Number of Residues5
DetailsBINDING SITE FOR RESIDUE SO4 A 1771
ChainResidue
AGLY539
ALYS540
ALYS618
AHOH2020
AHOH2077

site_idBC2
Number of Residues4
DetailsBINDING SITE FOR RESIDUE SO4 A 1772
ChainResidue
AARG470
ALYS618
AHIS679
AHOH2004

Functional Information from PROSITE/UniProt
site_idPS00107
Number of Residues31
DetailsPROTEIN_KINASE_ATP Protein kinases ATP-binding region signature. LGEGAFGQVVlAeaigldkdkpnrvtk...VAVK
ChainResidueDetails
ALEU484-LYS514

site_idPS00109
Number of Residues13
DetailsPROTEIN_KINASE_TYR Tyrosine protein kinases specific active-site signature. CIHrDLAARNVLV
ChainResidueDetails
ACYS619-VAL631

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PDB entries from 2024-10-09

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