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4TUU

Isolated p110a subunit of PI3Ka provides a platform for structure-based drug design

Functional Information from GO Data
ChainGOidnamespacecontents
A0016301molecular_functionkinase activity
A0046854biological_processphosphatidylinositol phosphate biosynthetic process
Functional Information from PROSITE/UniProt
site_idPS00915
Number of Residues15
DetailsPI3_4_KINASE_1 Phosphatidylinositol 3- and 4-kinases signature 1. FKng.DDLRQDmltlQ
ChainResidueDetails
APHE801-GLN815

site_idPS00916
Number of Residues21
DetailsPI3_4_KINASE_2 Phosphatidylinositol 3- and 4-kinases signature 2. ScAgycVatFILgIgDRHnsN
ChainResidueDetails
ASER900-ASN920

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsSITE: Implicated in the recognition of ATP as well as PIP2. Also crucial for autophosphorylation of the p85alpha subunit => ECO:0000305|PubMed:23936502
ChainResidueDetails
ALYS776

217705

PDB entries from 2024-03-27

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