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4PY4

Crystal structure of human poly(ADP-ribose) polymerase 14, catalytic domain in complex with an inhibitor XL2

Functional Information from GO Data
ChainGOidnamespacecontents
A0003950molecular_functionNAD+-protein poly-ADP-ribosyltransferase activity
B0003950molecular_functionNAD+-protein poly-ADP-ribosyltransferase activity
Functional Information from PDB Data
site_idAC1
Number of Residues9
DetailsBINDING SITE FOR RESIDUE XL2 A 1901
ChainResidue
AHIS1682
AGLY1683
ATYR1714
AALA1716
ATYR1721
ASER1722
ATYR1727
AGLN1764
APRO1766

site_idAC2
Number of Residues11
DetailsBINDING SITE FOR RESIDUE XL2 B 1901
ChainResidue
ASER1625
BHIS1682
BGLY1683
BASP1685
BTYR1701
BTYR1714
BTYR1721
BSER1722
BTHR1726
BTYR1727
BHOH2003

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PDB entries from 2024-10-09

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