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4P6X

Crystal Structure of cortisol-bound glucocorticoid receptor ligand binding domain

Functional Information from PDB Data
site_idAC1
Number of Residues12
Detailsbinding site for residue HCY A 900
ChainResidue
ALEU563
ATHR739
AILE747
AHOH1016
AASN564
AGLN570
AMET604
AARG611
APHE623
AGLN642
ATYR735
ACYS736

site_idAC2
Number of Residues12
Detailsbinding site for residue HCY C 900
ChainResidue
CLEU563
CASN564
CGLN570
CMET604
CARG611
CPHE623
CGLN642
CTYR735
CCYS736
CTHR739
CILE747
CHOH1010

site_idAC3
Number of Residues11
Detailsbinding site for residue HCY E 900
ChainResidue
ELEU563
EASN564
EGLN570
EARG611
EPHE623
EGLN642
ETYR735
ECYS736
ETHR739
EILE747
EHOH1059

site_idAC4
Number of Residues11
Detailsbinding site for residue HCY G 900
ChainResidue
GLEU563
GASN564
GGLN570
GMET604
GARG611
GPHE623
GGLN642
GTYR735
GCYS736
GTHR739
GILE747

site_idAC5
Number of Residues11
Detailsbinding site for residue HCY I 900
ChainResidue
ILEU563
IASN564
IGLN570
IMET604
IARG611
IPHE623
IGLN642
ITYR735
ICYS736
ITHR739
IILE747

site_idAC6
Number of Residues12
Detailsbinding site for residue HCY K 900
ChainResidue
KLEU563
KASN564
KGLN570
KMET604
KARG611
KPHE623
KGLN642
KTYR735
KCYS736
KTHR739
KILE747
KHOH1029

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues12
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO) => ECO:0000269|PubMed:12144530
ChainResidueDetails
ALYS703
KLYS703
CLYS703
ELYS703
GLYS703
ILYS703

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PDB entries from 2024-07-24

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