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4OJR

Crystal Structure of the HIV-1 Integrase catalytic domain with GSK1264

Functional Information from GO Data
ChainGOidnamespacecontents
A0003676molecular_functionnucleic acid binding
A0015074biological_processDNA integration
Functional Information from PDB Data
site_idAC1
Number of Residues12
DetailsBINDING SITE FOR RESIDUE 2SQ A 301
ChainResidue
AGLN95
AHIS171
ATHR174
AHOH452
ALEU102
ATHR125
AALA128
AALA129
ATRP132
AGLN168
AALA169
AGLU170

site_idAC2
Number of Residues4
DetailsBINDING SITE FOR RESIDUE CAC A 302
ChainResidue
ACYS65
AGLU92
ATHR97
AASN120

site_idAC3
Number of Residues4
DetailsBINDING SITE FOR RESIDUE CAC A 303
ChainResidue
ACYS130
AILE135
ALYS136
AGLN137

site_idAC4
Number of Residues7
DetailsBINDING SITE FOR RESIDUE SO4 A 304
ChainResidue
ALYS71
AARG166
AGLU170
AHIS171
ALEU172
AHOH409
AHOH497

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsBINDING: BINDING => ECO:0000250
ChainResidueDetails
AASP64
AASP116

site_idSWS_FT_FI2
Number of Residues1
DetailsBINDING: BINDING => ECO:0000250|UniProtKB:P04585
ChainResidueDetails
AGLU152

221371

PDB entries from 2024-06-19

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