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4MR6

Crystal Structure of the second bromodomain of human BRD2 in complex with a quinazolinone ligand (RVX-208)

Functional Information from PDB Data
site_idAC1
Number of Residues7
DetailsBINDING SITE FOR RESIDUE EDO A 501
ChainResidue
ATYR368
ALYS402
AASP407
AGLU413
AMET438
ALYS441
AHOH616

site_idAC2
Number of Residues7
DetailsBINDING SITE FOR RESIDUE EDO A 502
ChainResidue
AGLN443
AASP444
AGLU447
APHE448
AHOH724
ATYR426
AARG440

site_idAC3
Number of Residues6
DetailsBINDING SITE FOR RESIDUE EDO A 503
ChainResidue
ALYS351
AASP385
ATYR428
APRO430
AHOH754
AHOH772

site_idAC4
Number of Residues5
DetailsBINDING SITE FOR RESIDUE DMS A 504
ChainResidue
ATRP370
AHIS433
AMET438
AHOH660
AHOH723

site_idAC5
Number of Residues11
DetailsBINDING SITE FOR RESIDUE 1K0 A 505
ChainResidue
ALYS351
ATRP370
APRO371
APHE372
AVAL376
ALEU381
ALEU383
AASN429
AHIS433
AHOH606
AHOH660

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFykpvDasalglhDYHdiIkhpMdlstVkrkmenrd..Yrdaqefaadvrl.MfsNCykY
ChainResidueDetails
AALA369-TYR428

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PDB entries from 2024-09-11

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