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4LSJ

Crystal Structure of the Glucocorticoid Receptor Ligand Binding Domain Bound to a Dibenzoxapine Sulfonamide

Functional Information from PDB Data
site_idAC1
Number of Residues13
DetailsBINDING SITE FOR RESIDUE LSJ A 801
ChainResidue
ALEU563
ATYR735
ACYS736
ATHR739
APHE749
AASN564
AGLN570
AMET601
AMET604
ALEU608
APHE623
AMET639
ALEU732

site_idAC2
Number of Residues7
DetailsBINDING SITE FOR RESIDUE LSJ A 802
ChainResidue
ALEU532
APRO582
AASN586
ALEU685
ATHR692
ATRP712
ATYR716

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO) => ECO:0000269|PubMed:12144530
ChainResidueDetails
ALYS703

222415

PDB entries from 2024-07-10

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