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4LSJ

Crystal Structure of the Glucocorticoid Receptor Ligand Binding Domain Bound to a Dibenzoxapine Sulfonamide

Functional Information from PDB Data
site_idAC1
Number of Residues13
DetailsBINDING SITE FOR RESIDUE LSJ A 801
ChainResidue
ALEU563
ATYR735
ACYS736
ATHR739
APHE749
AASN564
AGLN570
AMET601
AMET604
ALEU608
APHE623
AMET639
ALEU732

site_idAC2
Number of Residues7
DetailsBINDING SITE FOR RESIDUE LSJ A 802
ChainResidue
ALEU532
APRO582
AASN586
ALEU685
ATHR692
ATRP712
ATYR716

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues165
DetailsRegion: {"description":"Interaction with CRY1","evidences":[{"source":"PubMed","id":"22170608","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

248636

PDB entries from 2026-02-04

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