4LSJ
Crystal Structure of the Glucocorticoid Receptor Ligand Binding Domain Bound to a Dibenzoxapine Sulfonamide
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 13 |
Details | BINDING SITE FOR RESIDUE LSJ A 801 |
Chain | Residue |
A | LEU563 |
A | TYR735 |
A | CYS736 |
A | THR739 |
A | PHE749 |
A | ASN564 |
A | GLN570 |
A | MET601 |
A | MET604 |
A | LEU608 |
A | PHE623 |
A | MET639 |
A | LEU732 |
site_id | AC2 |
Number of Residues | 7 |
Details | BINDING SITE FOR RESIDUE LSJ A 802 |
Chain | Residue |
A | LEU532 |
A | PRO582 |
A | ASN586 |
A | LEU685 |
A | THR692 |
A | TRP712 |
A | TYR716 |
Functional Information from SwissProt/UniProt
site_id | SWS_FT_FI1 |
Number of Residues | 2 |
Details | CROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO) => ECO:0000269|PubMed:12144530 |
Chain | Residue | Details |
A | LYS703 |