4LSJ
Crystal Structure of the Glucocorticoid Receptor Ligand Binding Domain Bound to a Dibenzoxapine Sulfonamide
Functional Information from PDB Data
| site_id | AC1 |
| Number of Residues | 13 |
| Details | BINDING SITE FOR RESIDUE LSJ A 801 |
| Chain | Residue |
| A | LEU563 |
| A | TYR735 |
| A | CYS736 |
| A | THR739 |
| A | PHE749 |
| A | ASN564 |
| A | GLN570 |
| A | MET601 |
| A | MET604 |
| A | LEU608 |
| A | PHE623 |
| A | MET639 |
| A | LEU732 |
| site_id | AC2 |
| Number of Residues | 7 |
| Details | BINDING SITE FOR RESIDUE LSJ A 802 |
| Chain | Residue |
| A | LEU532 |
| A | PRO582 |
| A | ASN586 |
| A | LEU685 |
| A | THR692 |
| A | TRP712 |
| A | TYR716 |
Functional Information from SwissProt/UniProt
| site_id | SWS_FT_FI1 |
| Number of Residues | 165 |
| Details | Region: {"description":"Interaction with CRY1","evidences":[{"source":"PubMed","id":"22170608","evidenceCode":"ECO:0000269"}]} |
| Chain | Residue | Details |






