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4L1A

Crystallographic study of multi-drug resistant HIV-1 protease Lopinavir complex: mechanism of drug recognition and resistance

Functional Information from GO Data
ChainGOidnamespacecontents
A0004190molecular_functionaspartic-type endopeptidase activity
A0006508biological_processproteolysis
B0004190molecular_functionaspartic-type endopeptidase activity
B0006508biological_processproteolysis
Functional Information from PDB Data
site_idAC1
Number of Residues22
DetailsBINDING SITE FOR RESIDUE AB1 A 101
ChainResidue
AARG8
AVAL84
AHOH223
AHOH245
AHOH247
AHOH259
AHOH309
BARG8
BASN25
BGLY27
BALA28
AASN25
BASP29
BGLY48
BPRO81
AGLY27
AALA28
AASP29
AASP30
AILE50
APRO81
ATHR82

237423

PDB entries from 2025-06-11

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