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4HNE

Crystal structure of the catalytic domain of human type II alpha Phosphatidylinositol 4-kinase (PI4KIIalpha) in complex with ADP

Functional Information from GO Data
ChainGOidnamespacecontents
A0004430molecular_function1-phosphatidylinositol 4-kinase activity
B0004430molecular_function1-phosphatidylinositol 4-kinase activity
Functional Information from PDB Data
site_idAC1
Number of Residues12
DetailsBINDING SITE FOR RESIDUE ADP A 500
ChainResidue
AGLY133
AILE345
AASP346
AHOH607
ASER134
ASER137
APHE139
ALYS152
AGLN261
ALEU262
APHE263
AVAL264

site_idAC2
Number of Residues8
DetailsBINDING SITE FOR RESIDUE ADP B 500
ChainResidue
BTYR131
BLYS152
BGLN261
BLEU262
BPHE263
BVAL264
BASP346
BHOH608

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues8
DetailsBINDING: BINDING => ECO:0000269|PubMed:24675427, ECO:0000269|PubMed:25168678
ChainResidueDetails
ATYR131
ALYS152
AGLN261
AASP346
BTYR131
BLYS152
BGLN261
BASP346

site_idSWS_FT_FI2
Number of Residues8
DetailsLIPID: S-palmitoyl cysteine => ECO:0000305|PubMed:22535966, ECO:0000305|PubMed:24675427
ChainResidueDetails
ASER174
ASER175
ASER177
ASER178
BSER174
BSER175
BSER177
BSER178

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PDB entries from 2024-04-24

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